Introducing

SIWA
318H™

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SIWA318H™:
A New Immunotherapy targeting Cancer and Aging-Related Diseases

SIWA Therapeutics has developed SIWA318H™, preparing to enter human clinical trials.

It targets cells damaged by oxidative stress, which is common in cancer and aging-related diseases.

SIWA318H™:
A Powerful New Treatment for Cancer and Aging Conditions

SIWA Therapeutics developed SIWA318H™, a humanized monoclonal antibody that targets a biomarker on cancer cells and other damaged/dysfunctional cells. SIWA318H™ works by stimulating the immune system’s ability to fight off harmful pathogens like bacteria, viruses, and cancer cells. The targeted biomarker indicates oxidative damage and is associated with cancer cells, as well as senescent cells, which play a key role in the development and progression of age-related diseases. Senescent cells also promote cancer progression and metastasis.

SIWA318H™ is an innovative immunotherapy that uses a dual-targeting mechanism to combat cancer and aging-related conditions.

SIWA318H™ targets diseased or dysfunctional cells to remove cells that cause or contribute to disease conditions. Its potential therapeutic benefits help with chronic kidney disease, osteoarthritis, aging related muscle wasting (sarcopenia), and infectious diseases. It has also shown effectiveness in targeting influenza and COVID-19-infected cells.

  • SIWA318H™ uses antibody-dependent cell-mediated cytotoxicity (ADCC) to target and eliminate cells with the oxidative stress marker. This marker is found on cancer cells, aging cells, and cells related to aging related diseases.
  • SIWA318H™ targets and eliminates cancer and aging cells. These cells can promote tumor growth and spread and weaken the immune system. Unlike traditional treatments, SIWA318H™ removes these cells from the tumor environment, improving the overall effectiveness of the therapy.
  • SIWA318H™ has shown effectiveness in targeting pancreatic cancer and glioblastoma cells, including those resistant to standard treatments, in preliminary studies conducted by TGen and the Illinois Institute of Technology Research Institute.
  • SIWA318H™ led to complete remission of pancreatic cancer in preclinical studies using immune-humanized mice. Treated groups showed significant tumor reduction, less severe disease, and increased survival compared to controls, without any adverse effects.
  • Additionally, in a Breast cancer model, a mouse version of SIWA318H™ reduced tumor growth and lung metastases.
  • Comprehensive Cancer Therapy: SIWA318H™ works by attacking both cancer cells and senescent cells. This dual approach weakens the tumor’s support network, which helps reduce cancer spread and growth. It may also lower the chances of cancer coming back. This strategy is especially important for aggressive cancers like pancreatic and breast cancer.
  • Anti-Aging and Regenerative Benefits : In addition to fighting cancer, SIWA318H™ also targets diseases related to aging e.g. by removing senescent cells. Tests in geriatric mice showed that SIWA318H™ increased the mass of muscles and reduced aging cells. This suggests it could help with weakness and age-related muscle loss (sarcopenia). The treatment has also shown promise against osteoarthritis and chronic kidney disease cells in human tissues.
  • Safe and Well-Tolerated: SIWA318H™ has shown no harmful side effects in various animal tests, including a tolerability study with non-human primates. This good safety record suggests it should be suitable for human clinical trials and eventual medical use.
  • The manufacturers can produce versions of the antibody for different animal species.
  • Unique Mechanism: Unlike treatments that turn cancer cells into senescent cells to stop cell division, SIWA318H™ actually removes both cancer cells and existing senescent cells. This is important because senescent cells can cause cancer to return, help new tumors form, and weaken the immune system.
  • No Interference with Co-Therapies: SIWA318H™ does not interfere with other treatments like CDK inhibitors (cancer drugs that affect cell division). Since it doesn’t interfere with these other treatments and is well-tolerated by the body, it’s a good option for combination approaches in both cancer treatment and regenerative medicine.
  • Potential for Orphan Drug Status: SIWA318H™ targets pancreatic cancer and other rare, aggressive cancers, so it may qualify as an “orphan drug” with the FDA.
  • This special status and possible fast-track designation could speed up its approval process and get it to patients sooner.

Conclusion

  • A Critical Investment Opportunity: Research shows SIWA318H™ could be a breakthrough treatment for both cancer and age-related diseases.
  • It works well, uses a unique approach, and can be used for many conditions. This makes its development and market launch important.
  • With no side effects observed and solid science behind it, SIWA318H™ could completely change how we treat cancer and approach regenerative medicine.

Credibility, Milestones, Significant Partnerships

Highlights of Worldwide Patent Portfolio

  • Patents have been granted to SIWA in Australia, China, Japan, Europe, Russia, South Korea, and the United States
  • All patents are owned by SIWA
  • SIWA has strong product and/or cancer therapy patent coverage in countries including the most important markets: North America, Europe and Asia
  • Patent prosecution is continuing with an eye toward expanded patent coverage

In February 2020, SIWA Therapeutics earned recognition as a “key player” in the Anti-Aging Drugs sector by MIT Technology Review, securing a place on its prestigious “10 Breakthrough Technologies of 2020” list.

TGen and SIWA318H™

TGen, the Translational Genomics Research Institute, a part of City of Hope, is an Arizona-based nonprofit that conducts groundbreaking medical research to improve lives.

TGen analyzes the genetic foundations of complex diseases, including cancer, neurological disorders, infectious diseases, and rare childhood conditions.

TGen received NIH grant funding to study the SIWA318H™ monoclonal antibody therapy in an advanced pancreatic cancer mouse model. The research evaluates the benefits of combining a mouse-compatible version of SIWA318H™ with current chemotherapy and immunotherapy treatments. 

The study is designed to demonstrate the value of the SIWA318H ™ antibody as an adjunct therapy for pancreatic cancer patients.

Charles River Laboratories

Charles River Laboratories accelerates research and drug development with essential products and services that transform possibilities into breakthroughs. From discovery through early development and safe manufacturing, they provide comprehensive solutions that help pharmaceutical, biotech, government, and academic teams bring new therapies to patients faster.

Founded in 1947 as a single laboratory in Boston overlooking the Charles River, it has grown into a global strategic partner with over 130 facilities across 20 countries. Our scientific expertise and comprehensive capabilities have contributed to over 80% of FDA-approved drugs in the past five years, establishing them as the partner of choice for nonclinical drug research and development.

Charles River Laboratories completed initial non-cGMP tolerability pharmacokinetic and toxicology studies of SIWA318H™ and tolerability assessments in both adult and juvenile non-human primates to support their FDA Investigational New Drug (IND) application.

Importantly, no adverse effects of the SIWA318H™ treatment were observed in any of these studies.

A DOCUMENTED HISTORY OF SUCCESS

Lewis Gruber
Misty Gruber
Dr. Gabriella Rossi, Ph.D

SIWA Therapeutics’ co-founders, Lewis and Misty Gruber, bring valuable experience in forming successful animal health partnerships. Their track record includes developing the commercially successful Sexcel technology through a collaboration between their previous venture and Genus ABS.

The Grubers have demonstrated a consistent ability to build strategic industry relationships, having earlier established a genomics partnership with American Cyanamid through another company they founded.

Complementing their business achievements, Misty Gruber has contributed to scientific knowledge in animal health through peer-reviewed research published in Poultry Science, adding academic credibility to their entrepreneurial expertise.

SIWA Therapeutics is led by a seasoned executive team with extensive industry expertise:
Lewis Gruber, Gabriela Rossi, Ph.D., and Misty Gruber.

Collectively, they bring over 75 years of experience in biotechnology and biopharmaceutical development to their leadership roles at SIWA.

Lewis Gruber
Director, Chief Executive Officer, and Chief Scientific Officer

Lewis Gruber co-founded SIWA Therapeutics after serving as director and interim CEO of a company that develops natural killer cell products. That research involves the natural killer cells that implement ADCC, which led to the actual SIWA318H technology.

 In 2000, Gruber co-founded Arryx, Inc., and served as its CEO until 2005, when it was acquired by a publicly traded company. Under his leadership, Arryx received prestigious recognitions, including the World Economic Forum Technology Pioneer award (2005), and was named among Red Herring’s Top 100 Innovators (2004).

From 1994 to 2000, Gruber was CEO and director of Hyseq, Inc., where he led the company through 1997’s largest biotech IPO and secured over $90 million in collaborative partnerships. He is the inventor of all SIWA intellectual property and has co-invented numerous other patented technologies.

In April 2020, Gruber was recognized on the Aging Analytics Agency’s list of 1000 Longevity Leaders. Before becoming an entrepreneur, he worked as a patent attorney specializing in biotechnology. He holds a J.D. and an M.S. in biology.

Contact: lsgruber@siwacorp.com

Misty Gruber co-founded SIWA Therapeutics after serving as a corporate finance expert at Dykema Gossett PLLC, where she was a member and Co-Chair of the biotechnology group. During her 29-year legal career, she represented various clients including issuers, investors, underwriters, and venture capital companies in transactions across North and South America, Europe, and Asia.

Beyond her legal expertise, Gruber was licensed as a CPA for several years, bringing valuable financial acumen to her role. She was also a co-founder of Arryx, Inc. and served as an initial director of Hyseq, Inc., demonstrating her long-standing involvement in biotechnology ventures.

Gruber holds a J.D., a B.S., and an M.S. in biology. In her leadership role at SIWA, she combines legal knowledge with scientific understanding.

Contact: msgruber@siwacorp.com

 

Misty Gruber
Director, Chief administrative Officer, and acting CFO
Gabriella Rossi
Chief Research Officer

Dr. Gabriela Rossi completed her undergraduate and doctoral education in Córdoba, Argentina, earning her Ph.D. in Infectious Disease and Immunology in 1997. Her distinguished postdoctoral training included fellowships at several prestigious institutions, including the National Institutes of Health (NIH), the National Cancer Institute, and the Iowa Cancer Research Foundation.

Throughout her career, Dr. Rossi has developed extensive expertise in immunology and diverse animal models used in biomedical research. Her scientific contributions have been published in peer-reviewed journals and presented at numerous national and international conferences.

Dr. Rossi brings valuable process development experience to SIWA Therapeutics, having worked with cGMP biological materials from early clinical trials through late-stage development. Her comprehensive background includes expertise in clinical study design and bridging laboratory research with therapeutic applications.

Contact: gabyrossi@siwacorp.com

 

Our Funding to Date

SIWA has adopted a model wherein we engage in contract and sponsored research work with top tier institutions such as TGen/City of Hope as well as with top Cancer Research Organizations. This model has allowed SIWA to retain all intellectual property rights while minimizing overhead. We believe this has allowed SIWA to be extremely efficient with our funds.

  • Pending completion of a Series B financing, we are funding SIWA through a $3,500,000 offering of Convertible Notes of which $3,000,000.00 of Note Principal was issued, with $500,000 remaining and available, which will convert at a discount into Series B Preferred Shares.
  • Altogether, we have raised approximately $11,100,000 (breakdown available upon request) in previous equity common, Series Seed, and Series A offerings, and the aforementioned convertible note offering. Our two principals are our largest investors by cash invested and shares held.